4-[2-(2-fluorophenoxymethyl)phenyl]piperidine compounds

US2016184288A1 · US · A1

Patent metadata
FieldValue
Publication numberUS-2016184288-A1
Application numberUS-201514848933-A
CountryUS
Kind codeA1
Filing dateSep 9, 2015
Priority dateNov 14, 2008
Publication dateJun 30, 2016
Grant date

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  1. Title

    What the patent document calls the invention.

  2. Abstract

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  3. Assignees and inventors

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  4. Key dates

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  5. First independent claim

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  6. CPC / IPC classifications

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  7. Citations and related patents

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Abstract

Official abstract text for this publication.

The invention relates to compounds of formula I: where a, R 1 , and R 3-6 are as defined in the specification, or a pharmaceutically acceptable salt thereof. The compounds of formula I are serotonin and norepinephrine reuptake inhibitors. The invention also relates to pharmaceutical compositions comprising such compounds; methods of using such compounds; and process and intermediates for preparing such compounds.

First claim

Opening claim text (preview).

What is claimed is: 1 . A pharmaceutical composition comprising a compound of the formula having the chemical name 4-[2-(2,4,6-trifluorophenoxymethyl)phenyl]piperidine or a pharmaceutically acceptable salt thereof and a pharmaceuticaly acceptable carrier. 2 . The pharmaceutical composition of claim 1 wherein the pharmaceutically acceptable salt is the hydrochloride salt. 3 . A method of treating a pain disorder in a mammal comprising administering to the mammal the pharmaceutical composition of claim 1 . 4 . The method of claim 3 wherein the pain disorder is neuropathic pain, fibromyalgia, chronic low back pain, or osteoarthritis.

Assignees

Inventors

Classifications

  • Drugs for disorders of the cardiovascular system · CPC title

  • Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives · CPC title

  • Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00 · CPC title

  • Antidepressants · CPC title

  • Anti-Parkinson drugs · CPC title

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Frequently asked questions

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What does patent US2016184288A1 cover?
The invention relates to compounds of formula I: where a, R 1 , and R 3-6 are as defined in the specification, or a pharmaceutically acceptable salt thereof. The compounds of formula I are serotonin and norepinephrine reuptake inhibitors. The invention also relates to pharmaceutical compositions compris…
Who is the assignee on this patent?
Patterson Lori Jean, Stangeland Eric L, Theravance Biopharma R&D Ip Llc
What technology area does this patent fall under?
Primary CPC classification A61K31/4465. Mapped technology areas include Human Necessities.
When was this patent published?
Publication date Thu Jun 30 2016 00:00:00 GMT+0000 (Coordinated Universal Time) (A1). Legal status and post-grant events are not shown on this page.
What related patents are in patentsdb?
We list 8 related publications on this page (citations in our corpus or others sharing the same primary CPC).