Pyrazole tetrahydronaphthyl carboxamides

Patent metadata

Field	Value
Publication number	US-9688608-B2
Application number	US-201514918729-A
Country	US
Kind code	B2
Filing date	Oct 21, 2015
Priority date	May 9, 2012
Publication date	Jun 27, 2017
Grant date	Jun 27, 2017

Abstract

The present invention relates to novel pyrazole(thio)tetrahydronaphthyl carboxamides, to processes for preparing these compounds, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms in crop protection and in the protection of materials.

First claim

The invention claimed is:

1. A Compound according to formula (III-a)

wherein
Q represents hydrogen;
X represents fluorine;
m represents 0 or 1;
R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 and R 8 independently from each other represent hydrogen or methyl;
wherein R 7 and R 8 can form the group ═C(Y 1 )Y 2 where Y 1 and Y 2 represent hydrogen or a group ═N—O—R c where R c represents methyl or ethyl,
and wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 and R 8 are not all hydrogen at the same time.

2. A compound according to claim 1 , wherein m is zero.

3. A compound according to claim 1 , wherein m is 1.

4. A compound according to claim 1 , wherein R 7 and R 8 form the group ═C(Y 1 )Y 2 .

5. A compound according to claim 1 , wherein R 7 and R 8 form the group ═N—O—R c .

6. A compound according to claim 1 , wherein at least one of R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 and R 8 is methyl.

7. A compound according to claim 1 , wherein at least two of R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 and R 8 are methyl.

8. A compound according to claim 5 , wherein R c represents methyl.

9. A compound according to claim 5 , wherein Rc represents ethyl.

Assignees

• Bayer Cropscience Ag

Inventors

• Maechling Simon
• Es-Sayed Mazen
• Dahmen Peter
• Wachendorff-Neumann Ulrike
• Bernier David
• Carles Lionel
• Dubost Christophe
• Vors Jean-Pierre
• Brunet Stephane
• Lachaise Helene

Classifications

• A01N43/56

  1,2-Diazoles; Hydrogenated 1,2-diazoles · CPC title

• C07D231/16 Primary

  Halogen atoms or nitro radicals · CPC title

• C07C2602/10

  the other ring being six-membered, e.g. tetraline · CPC title

• C07C211/60 Primary

  containing a ring other than a six-membered aromatic ring forming part of at least one of the condensed ring systems · CPC title

• C07C251/50

  having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals · CPC title