Besylate salt of a BTK inhibitor

US9604936B2 · US · B2

Patent metadata
FieldValue
Publication numberUS-9604936-B2
Application numberUS-201314058847-A
CountryUS
Kind codeB2
Filing dateOct 21, 2013
Priority dateAug 10, 2010
Publication dateMar 28, 2017
Grant dateMar 28, 2017

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  1. Title

    What the patent document calls the invention.

  2. Abstract

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  3. Assignees and inventors

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  4. Key dates

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  5. First independent claim

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  6. CPC / IPC classifications

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  7. Citations and related patents

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Abstract

Official abstract text for this publication.

The present invention provides a salt form, and compositions thereof, useful as an inhibitor of one or more protein kinases and which exhibits desirable characteristics for the same.

First claim

Opening claim text (preview).

We claim: 1. Compound 2: 2. The compound according to claim 1 , wherein said compound is in solid form. 3. The compound according to claim 2 , wherein said compound is crystalline. 4. The compound according to claim 3 , wherein said compound is a crystalline solid substantially free of amorphous Compound 2. 5. The compound according to claim 1 , wherein said compound is substantially free of impurities. 6. A composition comprising the compound according to claim 1 and a pharmaceutically acceptable carrier or excipient. 7. The compound according to claim 2 , wherein the solid form of the compound is characterized by at least one peak selected from the Form P1PXRD spectra depicted in FIG. 2 . 8. The compound according to claim 7 , wherein the solid form of the compound is characterized by at least two peaks selected from the Form P1PXRD spectra depicted in FIG. 2 . 9. The compound according to claim 8 , wherein the solid form of the compound is characterized by at least three peaks selected from the Form P1PXRD spectra depicted in FIG. 2 . 10. The compound according to claim 9 , wherein the solid form of the compound is characterized by at least four peaks selected from the Form P1PXRD spectra depicted in FIG. 2 . 11. The compound according to claim 2 , wherein the solid form of the compound is characterized by at least one peak selected from the Form P22PXRD spectra depicted in FIG. 6 . 12. The compound according to claim 11 , wherein the solid form of the compound is characterized by at least two peaks selected from the Form P22PXRD spectra depicted in FIG. 6 . 13. The compound according to claim 12 , wherein the solid form of the compound is characterized by at least three peaks selected from the Form P22PXRD spectra depicted in FIG. 6 . 14. The compound according to claim 13 , wherein the solid form of the compound is characterized by at least four peaks selected from the Form P22PXRD spectra depicted in FIG. 6 .

Assignees

Inventors

Classifications

  • Drugs for immunological or allergic disorders · CPC title

  • for hyperglycaemia, e.g. antidiabetics · CPC title

  • specific for metastasis · CPC title

  • Immunosuppressants, e.g. drugs for graft rejection · CPC title

  • Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors · CPC title

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Frequently asked questions

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What does patent US9604936B2 cover?
The present invention provides a salt form, and compositions thereof, useful as an inhibitor of one or more protein kinases and which exhibits desirable characteristics for the same.
Who is the assignee on this patent?
Celgene Avilomics Res Inc, Celgene Car Llc
What technology area does this patent fall under?
Primary CPC classification C07D239/48. Mapped technology areas include Chemistry & Metallurgy.
When was this patent published?
Publication date Tue Mar 28 2017 00:00:00 GMT+0000 (Coordinated Universal Time) (B2). Legal status and post-grant events are not shown on this page.
What related patents are in patentsdb?
We list 3 related publications on this page (citations in our corpus or others sharing the same primary CPC).