Aryloxyurea compound and pest control agent

Patent metadata

Field	Value
Publication number	US-9580384-B2
Application number	US-201514676921-A
Country	US
Kind code	B2
Filing date	Apr 2, 2015
Priority date	Oct 12, 2010
Publication date	Feb 28, 2017
Grant date	Feb 28, 2017

Abstract

The present invention provides a pest control agent, acaricide or fungicide that contains, as the active ingredient thereof, at least one type of compound selected from the aryloxyurea compounds represented by formula (V) (wherein R 1 to R 5 each independently represents an alkyl group or the like, X is a halogen atom or the like, n is an integer of 0 to 5, and Z is an oxygen atom or sulfur atom) or salts thereof.

First claim

The invention claimed is:

1. An aryloxyurea compound of formula (I) or a salt thereof:

wherein in formula (I), Cy is a C6-10 aryl group;
X is an unsubstituted or substituted C1-6 alkyl group, unsubstituted or substituted C3-8 cycloalkyl group, unsubstituted or substituted C2-6 alkenyl group, unsubstituted or substituted C2-6 alkynyl group, hydroxy group, unsubstituted or substituted C1-6 alkoxy group, amino group, unsubstituted or substituted C1-6 alkyl amino group, unsubstituted or substituted C1-7 acyl group, unsubstituted or substituted C1-6 alkoxycarbonyl group, unsubstituted or substituted C1-6 alkyl sulfonyl group, unsubstituted or substituted C1-6 alkoxysulfonyl group, unsubstituted or substituted C6-10 aryl group, unsubstituted or substituted heteroaryl group, unsubstituted or substituted hydroxyimino C1-6 alkyl group, nitro group, cyano group, or halogen atom;
n is the number of X bonded to Cy and is an integer of 0 to 5; when n is 2 or more, X may be mutually the same or different, and when n is 2 or more, X may bond together to form a ring together with the carbon atoms or nitrogen atoms bonded thereto;
R 1 is an unsubstituted or substituted C1-6 alkyl group, unsubstituted or substituted C2-6 alkenyl group, or unsubstituted or substituted C2-6 alkynyl group, wherein R 1 is not an unsubstituted or substituted C1-7 acyl group;
Q is a group of formula (II):

wherein in formula (II),
* is the bonding position;
R 2 is a hydrogen atom, unsubstituted or substituted C1-6 alkyl group, unsubstituted or substituted C2-6 alkenyl group, unsubstituted or substituted C2-6 alkynyl group, unsubstituted or substituted C1-7 acyl group, or unsubstituted or substituted C1-6 alkoxycarbonyl group, R 1 and R 2 may bond together to form an unsubstituted or substituted C2-4 alkylene group;
R 3 and R 4 each independently is an unsubstituted or substituted C1-6 alkyl group;
R 5 is an unsubstituted or substituted C6-10 aryl group, unsubstituted or substituted heteroaryl group, or unsubstituted or substituted aminocarbonyl group;
Z is an oxygen atom or sulfur atom.

2. A pest control agent, comprising at least one of the aryloxyurea compound or a salt thereof according to claim 1 as an active ingredient.

3. An acaricide, comprising at least one of the aryloxyurea compound or a salt thereof according to claim 1 as an active ingredient.

4. An aryloxyurea compound of formula (I) or a salt thereof:

wherein in formula (I), Cy is a heteroaryl aryl group;
X is an unsubstituted or substituted C1-6 alkyl group, unsubstituted or substituted C3-8 cycloalkyl group, unsubstituted or substituted C2-6 alkenyl group, unsubstituted or substituted C2-6 alkynyl group, hydroxy group, unsubstituted or substituted C1-6 alkoxy group, amino group, unsubstituted or substituted C1-6 alkyl amino group, unsubstituted or substituted C1-7 acyl group, unsubstituted or substituted C1-6 alkoxycarbonyl group, unsubstituted or substituted C1-6 alkyl sulfonyl group, unsubstituted or substituted C1-6 alkoxysulfonyl group, unsubstituted or substituted C6-10 aryl group, unsubstituted or substituted heteroaryl group, unsubstituted or substituted hydroxyimino C1-6 alkyl group, nitro group, cyano group, or halogen atom;
n is the number of X bonded to Cy and is an integer of 0 to 5; when n is 2 or more, X may be mutually the same or different, and when n is 2 or more, X may bond together to form a ring together with the carbon atoms or nitrogen atoms bonded thereto;
R 1 is an unsubstituted or substituted C1-6 alkyl group, unsubstituted or substituted C2-6 alkenyl group, or unsubstituted or substituted C2-6 alkynyl group, wherein R 1 is not an unsubstituted or substituted C1-7 acyl group;
Q is a group of formula (II):

wherein in formula (II),
* is the bonding position;
R 2 is a hydrogen atom, unsubstituted or substituted C1-6 alkyl group, unsubstituted or substituted C2-6 alkenyl group, unsubstituted or substituted C2-6 alkynyl group, unsubstituted or substituted C1-7 acyl group, or unsubstituted or substituted C1-6 alkoxycarbonyl group, R 1 and R 2 may bond together to form an unsubstituted or substituted C2-4 alkylene group;
R 3 and R 4 each independently is an unsubstituted or substituted C1-6 alkyl group;
R 5 is an unsubstituted or substituted aminocarbonyl group;
Z is an oxygen atom or sulfur atom.

Assignees

• Nippon Soda Co

Inventors

• Furukawa Hironori
• Nakamura Takehiko
• Tamai Tetsuo
• Hanai Daisuke

Classifications

• A01N47/32

  containing >N—CO—N< or >N—CS—N< groups directly attached to a cycloaliphatic ring · CPC title

• C07D213/74

  Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals · CPC title

• C07D253/065

  having three double bonds between ring members or between ring members and non-ring members · CPC title

• A61K31/4418

  having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine · CPC title

• C07D239/26

  with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms · CPC title