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Nitrogen-containing aromatic heterocyclyl compound
US9150563B2 · US · B2
| Field | Value |
|---|---|
| Publication number | US-9150563-B2 |
| Application number | US-201414177000-A |
| Country | US |
| Kind code | B2 |
| Filing date | Feb 10, 2014 |
| Priority date | Jul 8, 2008 |
| Publication date | Oct 6, 2015 |
| Grant date | Oct 6, 2015 |
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Abstract
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The present invention provides a compound having excellent regulating action on blood lipid level. The present invention provides a compound represented by the following general formula (I) or a pharmacologically acceptable salt thereof, etc., wherein A represents a 5-membered nitrogen-containing aromatic heterocyclyl group; R 1 represents COOH or the like; each R 2 represents an alkyl or the like; each R 3 represents an optionally substituted phenyl, an optionally substituted phenylalkyl, or the like; m represents 0, 1, 2, or 3; n represents 0 or 1; each of R 4 , R 5 , R 6 , and R 7 represents H, an alkyl, or the like; and B represents an optionally substituted naphthyl, an optionally substituted aromatic heterocyclyl, or a group represented by the following formula (II) wherein each of B 1 and B 2 represents an optionally substituted phenyl or an optionally substituted aromatic heterocyclyl.
First claim
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The invention claimed is: 1. 4-{3-[2-(4-Hydroxyphenyl)thiazol-5-yl]-2-fluoropropanoyl}amino-1-ethylpyrrole-3-carboxylic acid or a pharmacologically acceptable salt thereof. 2. A method for the treatment of a disease selected from hyperlipidemia, dyslipidemia, lipid metabolism abnormality, arteriosclerosis, hypertriglyceridemia, non-alcoholic steatohepatitis, or type II diabetes mellitus, which comprises administering a pharmaceutically effective amount of the co…
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Frequently asked questions
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- What does patent US9150563B2 cover?
- The present invention provides a compound having excellent regulating action on blood lipid level. The present invention provides a compound represented by the following general formula (I) or a pharmacologically acceptable salt thereof, etc., wherein A represents a 5-membered nitrogen-containing aromatic heterocyclyl group; R 1 represents COOH or the like; each R 2 represents an alkyl …
- Who is the assignee on this patent?
- Daiichi Sankyo Co Ltd
- What technology area does this patent fall under?
- Primary CPC classification C07D417/12. Mapped technology areas include Chemistry & Metallurgy.
- When was this patent published?
- Publication date Tue Oct 06 2015 00:00:00 GMT+0000 (Coordinated Universal Time) (B2). Legal status and post-grant events are not shown on this page.
- What related patents are in patentsdb?
- We list 8 related publications on this page (citations in our corpus or others sharing the same primary CPC).