Androgen receptor modulators and uses thereof

Patent metadata

Field	Value
Publication number	US-9108944-B2
Application number	US-201113579009-A
Country	US
Kind code	B2
Filing date	Feb 16, 2011
Priority date	Feb 16, 2010
Publication date	Aug 18, 2015
Grant date	Aug 18, 2015

Abstract

Described herein are compounds that are androgen receptor modulators. Also described are pharmaceutical compositions and medicaments that include the compounds described herein, as well as methods of using such androgen receptor modulators, alone and in combination with other compounds, for treating diseases or conditions that are mediated or dependent upon androgen receptors.

First claim

What is claimed is:

1. A compound of Formula (Ia), or a pharmaceutically acceptable salt, or N-oxide thereof:

wherein,
ring A is pyridinyl;
m is 1, 2, 3 or 4;
each R A is independently halogen, —CN, —NO 2 , —OH, —OR 9 , —SR 9 , —S(═O)R 10 , —S(═O) 2 R 10 , —N(R 11 )S(═O) 2 R 10 , —S(═O) 2 N(R 9 ) 2 , —C(═O)R 10 , —OC(═O)R 10 , —CO 2 R 9 , —N(R 9 )…

Assignees

• Smith Nicholas D
• Bonnefous Celine
• Julien Jackaline D
• Aragon Pharmaceuticals Inc

Inventors

• Smith Nicholas D
• Bonnefous Celine
• Julien Jackaline D

Classifications

• A61P9/00

  Human Necessities · mapped topic

• A61P9/10

  Human Necessities · mapped topic

• A61P5/28

  Human Necessities · mapped topic

• A61P35/00

  Human Necessities · mapped topic

• A61P5/26

  Human Necessities · mapped topic