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US8999994B2 · US · B2
| Field | Value |
|---|---|
| Publication number | US-8999994-B2 |
| Application number | US-201113635894-A |
| Country | US |
| Kind code | B2 |
| Filing date | Mar 18, 2011 |
| Priority date | Mar 18, 2010 |
| Publication date | Apr 7, 2015 |
| Grant date | Apr 7, 2015 |
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- Title
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- Abstract
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Abstract
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The present invention relates to a compound of formula (I): wherein: R 1 and R 2 are selected from among H and C1-C10 alkyl; R 3 is selected from among H, —OR 4 , N, —CN, —C(O)R 4 , —C(O)OR 4 , —C(O)NR 4 R 5 , —C═NR 4 , —OC(O)R 4 , —NR 4 R 5 , —NR 4 C(O)R 5 , —NO 2 , —N═CR 4 R 5 , halogen and C1-C10 alkyl, wherein R 4 and R 5 are selected from among H, alkyl, alkenyl, cycloalkyl and aryl; X, Y, Z 1 , Z 2 and Z 3 are selected independently from among CH and N; A is selected from among (CH 2 ) n , NH, O and CO, wherein n is an integer between 1 and 6, to the procedure for the obtainment of said compounds, to a pharmaceutical composition comprising said compound, and to the use thereof in the treatment of a neurodegenerative disease, more particularly treatment of Alzheimer's or Parkinson's disease.
First claim
Opening claim text (preview).
The invention claimed is: 1. A compound of formula (I) where, R 1 and R 2 are selected from H and C 1 -C 10 alkyl, R 3 is selected from H, —OR 4 , N, —CN, —C(O)R 4 , —C(O)OR 4 , —C(O)NR 4 R 5 , —C═NR 4 , —OC(O)R 4 , —NR 4 R 5 , —NR 4 C(O)R 5 , —NO 2 , —N═CR 4 R 5 , halogen and C 1 -C 10 alkyl, where R 4 and R 5 are selected from H, alkyl, alkenyl, cycloalkyl a…
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Human Necessities · mapped topic
Chemistry & Metallurgy · mapped topic
- C07D401/12Primary
Chemistry & Metallurgy · mapped topic
Human Necessities · mapped topic
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- What does patent US8999994B2 cover?
- The present invention relates to a compound of formula (I): wherein: R 1 and R 2 are selected from among H and C1-C10 alkyl; R 3 is selected from among H, —OR 4 , N, —CN, —C(O)R 4 , —C(O)OR 4 , —C(O)NR 4 R 5 , —C═NR 4 , —OC(O)R 4 , —NR 4 R 5 , —NR 4 C(O)R 5 , —NO 2 , —N═CR 4 R 5 , halogen and C1-C10 a…
- Who is the assignee on this patent?
- Samadi Abdelouahid, Marco Contelles José Luis, Bolea Tomás Irene, and 5 more
- What technology area does this patent fall under?
- Primary CPC classification C07D401/12. Mapped technology areas include Chemistry & Metallurgy.
- When was this patent published?
- Publication date Tue Apr 07 2015 00:00:00 GMT+0000 (Coordinated Universal Time) (B2). Legal status and post-grant events are not shown on this page.
- What related patents are in patentsdb?
- We list 8 related publications on this page (citations in our corpus or others sharing the same primary CPC).