Boron-containing pharmacophore

US12065456B2 · US · B2

Patent metadata
FieldValue
Publication numberUS-12065456-B2
Application numberUS-202016881272-A
CountryUS
Kind codeB2
Filing dateMay 22, 2020
Priority dateJul 25, 2019
Publication dateAug 20, 2024
Grant dateAug 20, 2024

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  1. Title

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  2. Abstract

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  3. Assignees and inventors

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  4. Key dates

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  5. First independent claim

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  6. CPC / IPC classifications

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  7. Citations and related patents

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Abstract

Official abstract text for this publication.

Provided herein are boron-containing compounds, pharmaceutical compositions comprising such compounds, and methods of using such compounds to treat diseases or disorders.

First claim

Opening claim text (preview).

The invention claimed is: 1. A compound of Formula Ia: or a pharmaceutically acceptable salt thereof; wherein B is boron; and W is absent or C(R 3 ) 2 ; and R 3 is independently, at each occurrence, selected from the group consisting of H, halo, C 1 -C 6 alkyl, C 1 -C 6 alkoxy, C 6 -C 10 aryl, C 5 -C 10 heteroaryl, C 3 -C 10 cycloalkyl, and C 3 -C 10 heterocycloalkyl. 2. The compound of claim 1 , wherein W is absent. 3. The compound of claim 1 , wherein W is CH 2 . 4. The compound of claim 1 , wherein W is C(R 3 ) 2 .

Assignees

Inventors

Classifications

  • C07F5/025Primary

    Boronic and borinic acid compounds · CPC title

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Frequently asked questions

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What does patent US12065456B2 cover?
Provided herein are boron-containing compounds, pharmaceutical compositions comprising such compounds, and methods of using such compounds to treat diseases or disorders.
Who is the assignee on this patent?
Massachusetts Inst Technology, Nat Institutes Of Health Nih U S Dept Of Health And Human Services Dhhs U S Government
What technology area does this patent fall under?
Primary CPC classification C07F5/025. Mapped technology areas include Chemistry & Metallurgy.
When was this patent published?
Publication date Tue Aug 20 2024 00:00:00 GMT+0000 (Coordinated Universal Time) (B2). Legal status and post-grant events are not shown on this page.
What related patents are in patentsdb?
We list 8 related publications on this page (citations in our corpus or others sharing the same primary CPC).