NRF2 activators

US11028099B2 · US · B2

Patent metadata
FieldValue
Publication numberUS-11028099-B2
Application numberUS-201716469203-A
CountryUS
Kind codeB2
Filing dateDec 11, 2017
Priority dateDec 15, 2016
Publication dateJun 8, 2021
Grant dateJun 8, 2021

How to read this patent

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  1. Title

    What the patent document calls the invention.

  2. Abstract

    A short plain-language summary of the technical disclosure.

  3. Assignees and inventors

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  4. Key dates

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  5. First independent claim

    The legal scope of protection — read this for what is actually claimed.

  6. CPC / IPC classifications

    Technology tags used to group this patent with similar filings.

  7. Citations and related patents

    Prior art links and similar publications in this corpus.

Abstract

Official abstract text for this publication.

The present invention relates to a compound which is (R)-3-(1,4-dimethyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(3-(((R)-2-ethyl-2,3-dihydropyrido[2,3-f][1,4]oxazepin-4(5H)-yl)methyl)-4-methylphenyl)propanoic acid (I), or a pharmaceutically acceptable salt thereof, in particular, the meglumine salt thereof, a pharmaceutical composition containing the compound and its use as an NRF2 activator.

First claim

Opening claim text (preview).

What is claimed is: 1. A compound which is (R)-3-(1,4-dimethyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(3-(((R)-2-ethyl-2,3-dihydropyrido[2,3-f][1,4]oxazepin-4(5H)-yl)methyl)-4-methylphenyl)propanoic acid: or a pharmaceutically acceptable salt thereof. 2. A pharmaceutical composition comprising the compound of claim 1 and one or more pharmaceutically acceptable excipients.

Assignees

Inventors

Classifications

  • of the kidneys · CPC title

  • Antineoplastic agents · CPC title

  • C07D498/04Primary

    Ortho-condensed systems · CPC title

  • Drugs for disorders of the cardiovascular system · CPC title

  • ortho- or peri-condensed with heterocyclic ring systems · CPC title

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Frequently asked questions

Answers are generated from the same data shown on this page.

What does patent US11028099B2 cover?
The present invention relates to a compound which is (R)-3-(1,4-dimethyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(3-(((R)-2-ethyl-2,3-dihydropyrido[2,3-f][1,4]oxazepin-4(5H)-yl)methyl)-4-methylphenyl)propanoic acid (I), or a pharmaceutically acceptable salt thereof, in particular, the meglumine salt thereof, a pharmaceutical composition containing the compound and its use as an NRF2 activator.
Who is the assignee on this patent?
Glaxosmithkline Ip Dev Ltd
What technology area does this patent fall under?
Primary CPC classification C07D498/04. Mapped technology areas include Chemistry & Metallurgy.
When was this patent published?
Publication date Tue Jun 08 2021 00:00:00 GMT+0000 (Coordinated Universal Time) (B2). Legal status and post-grant events are not shown on this page.
What related patents are in patentsdb?
We list 2 related publications on this page (citations in our corpus or others sharing the same primary CPC).