Heterocyclic compounds as pesticides

Patent metadata

Field	Value
Publication number	US-10961201-B2
Application number	US-201916536902-A
Country	US
Kind code	B2
Filing date	Aug 9, 2019
Priority date	Oct 2, 2012
Publication date	Mar 30, 2021
Grant date	Mar 30, 2021

Abstract

The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds.

First claim

The invention claimed is:

1. A method for controlling one or more pests, comprising allowing a compound of formula (I)

to act on one or more pests and/or a habitat thereof,
in which
A represents

 in which the broken line represents the bond to Q and in which A furthermore carries m substituents R2,
Q represents a radical Q-2

 in which the nitrogen is attached to ring A and the arrow in each case represents the bond to D and
D represents the radical of the formula

 in which the nitrogen is attached to Q and the arrow represents the bond to B,
B represents

 in which the broken line the bond to D and in which B furthermore carries n substituents R7,
Z represents oxygen or sulphur,
R1 represents a radical from the group consisting of halogen, cyano, nitro, amino, hydroxy, represents C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -alkenyloxy, C 3 -C 6 -alkynyloxy, C 3 -C 6 -cycloalkyloxy, C 1 -C 6 -alkylcarbonyloxy, C 2 -C 6 -alkenylcarbonyloxy, C 2 -C 6 -alkynylcarbonyloxy, C 3 -C 6 -cycloalkylcarbonyloxy, C 1 -C 6 -alkoxycarbonyloxy, C 1 -C 6 -alkylsulphonyloxy, C 1 -C 6 -alkylamino, C 3 -C 6 -alkenylamino, C 3 -C 6 -alkynylamino, C 3 -C 6 -cycloalkylamino, C 1 -C 6 -alkylcarbonylamino, C 2 -C 6 -alkenylcarbonylamino, C 2 -C 6 -alkynylcarbonylamino, C 3 -C 6 -cycloalkylcarbonylamino, C 1 -C 6 -alkoxycarbonylamino, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylthio, C 3 -C 6 -alkenylthio, C 3 -C 6 -alkynylthio, C 3 -C 6 -cycloalkylthio, C 1 -C 6 -alkylsulphinyl, C 1 -C 6 -alkylsulphonyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxyimino-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl, aminocarbonyl, C 1 -C 6 -alkylaminocarbonyl, di-(C 1 -C 6 -alkyl)-aminocarbonyl, aminothiocarbonyl, C 1 -C 6 -alkylaminosulphonyl, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylcarbonylamino, C 1 -C 6 -alkylthiocarbonylamino, C 4 -C 12 — bicycloalkyl, aryl, aryloxy, arylamino, and arylthio, each of which is optionally substituted by one or more identical or different substituents, where the substituents independently of one another are selected from the group consisting of halogen, cyano, nitro, hydroxy, amino, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, aryl, aryloxy, and arylthio,
R2 represents a radical from the group consisting of halogen, cyano, nitro, amino, hydroxy, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -alkenoxy, C 3 -C 6 -alkynoxy, C 3 -C 6 -cycloalkoxy, C 1 -C 6 -alkylcarbonyloxy, C 2 -C 6 -alkenylcarbonyloxy, C 2 -C 6 -alkynylcarbonyloxy, C 3 -C 6 -cycloalkylcarbonyloxy, C 1 -C 6 -alkoxycarbonyloxy, C 1 -C 6 -alkylsulphonyloxy, C 1 -C 6 -alkylamino, di-(C 1 -C 6 -alkyl)-amino, C 1 -C 6 -alkenylamino, C 3 -C 6 -alkynylamino, C 3 -C 6 -cycloalkylamino, C 3 -C 6 -alkylcarbonylamino, C 1 -C 6 -alkenylcarbonylamino, C 2 -C 6 -alkynylcarbonylamino, C 3 -C 6 -cycloalkylcarbonylamino, C 1 -C 6 -alkoxycarbonylamino, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylthio, C 3 -C 6 -alkenylthio, C 3 -C 6 -alkynylthio, C 3 -C 6 -cycloalkylthio, C 1 -C 6 -alkylsulphinyl, C 1 -C 6 -alkylsulphonyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxyimino-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl, aminocarbonyl, C 1 -C 6 -alkylaminocarbonyl, di-(C 1 -C 6 -alkyl)-aminocarbonyl, aminothiocarbonyl, C 1 -C 6 -alkylaminosulphonyl, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylcarbonylamino, C 1 -C 6 -alkylthiocarbonylamino, C 4 -C 12 -bicycloalkyl, aryl, aryloxy, arylamino, and arylthio, each of which is optionally substituted by one or more identical or different substituents, where the substituents independently of one another are selected from the group consisting of halogen, cyano, nitro, hydroxy, amino, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, C 1 -C 6 -haloalkoxy and C 1 -C 6 -alkylthio, aryl, aryloxy, and arylthio,
R3 represents a radical from the group consisting of hydrogen, halogen, cyano, nitro, amino, hydroxy, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkyl and C 1 -C 6 -haloalkoxy,
R5 represents a radical from the group consisting of hydrogen, C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -haloalkyl, C 2 -C 6 -alkenyl, C 3 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkyl, cyano-C 1 -C 6 -alkyl, C 1 -C 6 -alkylcarbonyl, C 2 -C 6 -alkenylcarbonyl, C 1 -C 6 -haloalkylcarbonyl, C 2 -C 6 -haloalkenylcarbonyl, C 1 -C 6 -alkoxy-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl, C 1 -C 6 -alkylsulphonyl and C 1 -C 6 -haloalkylsulphonyl or represents C(═O)—B,
R6 represents a radical from the group consisting of halogen, cyano, nitro, amino, hydroxy, carboxyl, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -alkenoxy, C 3 -C 6 -alkynoxy, C 3 -C 6 -cycloalkoxy, C 1 -C 6 -alkylcarbonyloxy, C 2 -C 6 -alkenylcarbonyloxy, C 2 -C 6 -alkynylcarbonyloxy, C 3 -C 6 -cycloalkylcarbonyloxy, C 1 -C 6 -alkoxycarbonyloxy, C 1 -C 6 -alkylsulphonyloxy, C 1 -C 6 -alkylcarbonylamino, C 2 -C 6 -alkenylcarbonylamino, C 2 -C 6 -alkynylcarbonylamino, C 3 -C 6 -cycloalkylcarbonylamino, C 1 -C 6 -alkoxycarbonylamino, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylthio, C 1 -C 6 -alkylsulphinyl, C 1 -C 6 -alkylsulphonyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxyimino-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl, aminocarbonyl, C 1 -C 6 -alkylaminocarbonyl, di-(C 1 -C 6 -alkyl)-aminocarbonyl, aminothiocarbonyl, C 1 -C 6 -alkylaminosulphonyl, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylcarbonylamino, C 1 -C 6 -haloalkylcarbonylamino, C 1 -C 6 -alkylthiocarbonylamino, C 4 -C 12 -bicycloalkyl, aryl, and aryloxy, each of which is optionally substituted by one or more identical or different substituents, where the substituents independently of one another are selected from the group consisting of halogen, cyano, nitro, hydroxy, amino, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, C 1 -C 6 -haloalkoxy and C 1 -C 6 -alkylthio,
R7 represents a radical from the group consisting of halogen, nitro, cyano, amino, hydroxy, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -alkenoxy, C 3 -C 6 -alkynoxy, C 3 -C 6 -cycloalkoxy, C 1 -C 6 -alkylcarbonyloxy, C 2 -C 6 -alkenylcarbonyloxy, C 2 -C 6 -alkynylcarbonyloxy, C 3 -C 6 -cycloalkylcarbonyloxy, C 1 -C 6 -alkoxycarbonyloxy, C 1 -C 6 -alkylsulphonyloxy, C 1 -C 6 -alkylcarbonylamino, C 2 -C 6 -alkenylcarbonylamino, C 2 -C 6 -alkynylcarbonylamino, C 3 -C 6 -cycloalkylcarbonylamino, C 1 -C 6 -alkoxycarbonylamino, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylthio, C 1 -C 6 -alkylsulphinyl, C 1 -C 6 -alkylsulphonyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxyimino-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl, aminocarbonyl, C 1 -C 6 -alkylaminocarbonyl, di-(C 1 -C 6 -alkyl)-aminocarbonyl, aminothiocarbonyl, C 1 -C 6 -alkylaminosulphonyl, C 1 -C 6 -alkylsulphonylamino, C 1 -C 6 -alkylcarbonylamino, C 1 -C 6 -alkylthiocarbonylamino, aryl, aryloxy, and C 4 -C 12 -bicycloalkyl, each of which is optionally substituted by one or more identical or different substituents, where the substituents independently of one another are selected from the group consisting of halogen, cyano, nitro, hydroxy, amino, C 1 -C 6 -alk

Assignees

• Bayer Cropscience Ag

Inventors

• Heilmann Eike Kevin
• Greul Joerg
• Trautwein Axel
• Schwarz Hans-Georg
• Adelt Isabelle
• Andree Roland
• Luemmen Peter
• Hink Maike
• Adamczewski Martin
• Drewes Mark
• Becker Angela
• Voerste Arnd
• Goergens Ulrich
• Ilg Kerstin
• Jansen Johannes-Rudolf
• Portz Daniela

Classifications

• C07D231/40 Primary

  Acylated on said nitrogen atom · CPC title

• C07D231/06

  having one double bond between ring members or between a ring member and a non-ring member · CPC title

• C07D403/12

  linked by a chain containing hetero atoms as chain links · CPC title

• A01N43/76

  1,3-Oxazoles; Hydrogenated 1,3-oxazoles · CPC title

• A61P33/00

  Antiparasitic agents · CPC title