Pharmaceutical formulations comprising a pyridylaminoacetic acid compound

US10179127B2 · US · B2

Patent metadata
FieldValue
Publication numberUS-10179127-B2
Application numberUS-201815895100-A
CountryUS
Kind codeB2
Filing dateFeb 13, 2018
Priority dateJan 10, 2014
Publication dateJan 15, 2019
Grant dateJan 15, 2019

How to read this patent

A practical reading order for non-experts. Skip the full description unless you need deep technical detail.

  1. Title

    What the patent document calls the invention.

  2. Abstract

    A short plain-language summary of the technical disclosure.

  3. Assignees and inventors

    Who owns or filed the patent and who is credited as inventor.

  4. Key dates

    Filing, priority, publication, and grant dates set the timeline.

  5. First independent claim

    The legal scope of protection — read this for what is actually claimed.

  6. CPC / IPC classifications

    Technology tags used to group this patent with similar filings.

  7. Citations and related patents

    Prior art links and similar publications in this corpus.

Abstract

Official abstract text for this publication.

Provided is a pharmaceutical preparation for treatment or prevention of glaucoma or ocular hypertension, comprising 0.0003 to 0.01% (w/v) of isopropyl (6-{[4-(pyrazol-1-yl)benzyl] (pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino) acetate, or a salt thereof. The pharmaceutical preparation has an excellent intraocular pressure lowering effect and may be used as a therapeutic or preventive agent for glaucoma or ocular hypertension or an intraocular pressure lowering agent.

First claim

Opening claim text (preview).

The invention claimed is: 1. A pharmaceutical preparation for treatment or prevention of glaucoma or ocular hypertension, comprising 0.002% (w/v) of isopropyl (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)acetate, or a salt thereof. 2. The pharmaceutical preparation according to claim 1 , in which the preparation is for treatment of glaucoma. 3. The pharmaceutical preparation according to claim 1 , in which the preparation is for treatment of ocular hypertension. 4. The pharmaceutical preparation according to claim 1 , in which the preparation does not include other therapeutic agents for glaucoma. 5. The pharmaceutical preparation according to claim 1 , in which the preparation is not used in combination with other therapeutic agents for glaucoma. 6. An eye drop comprising the pharmaceutical preparation of claim 1 . 7. A method for treatment or prevention of glaucoma or ocular hypertension, comprising administrating the pharmaceutical preparation of claim 1 to a patient who needs the treatment or prevention of glaucoma or ocular hypertension. 8. A method for treatment of glaucoma, comprising administrating the pharmaceutical preparation of claim 2 to a patient who needs the treatment of glaucoma. 9. A method for treatment of ocular hypertension, comprising administrating the pharmaceutical preparation of claim 3 to a patient who needs the treatment of ocular hypertension. 10. The method of claim 7 , in which the preparation does not include other therapeutic agents for glaucoma. 11. The method of claim 7 , the preparation is not used in combination with other therapeutic agents for glaucoma. 12. The method of claim 7 , in which the administrating is instillation. 13. The method of claim 12 , in which the instillation is provided once or twice a day. 14. The method of claim 7 , in which a dose of one or two drops is instilled. 15. The method of claim 7 , in which a dose of one drop is instilled once a day. 16. The method of claim 7 , wherein the patient is a human.

Assignees

Inventors

Classifications

  • Ophthalmic agents · CPC title

  • A61K31/444Primary

    containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone · CPC title

  • Eye, e.g. artificial tears · CPC title

  • Antiglaucoma agents or miotics · CPC title

Patent family

Related publications grouped by family.

External sources

Frequently asked questions

Answers are generated from the same data shown on this page.

What does patent US10179127B2 cover?
Provided is a pharmaceutical preparation for treatment or prevention of glaucoma or ocular hypertension, comprising 0.0003 to 0.01% (w/v) of isopropyl (6-{[4-(pyrazol-1-yl)benzyl] (pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino) acetate, or a salt thereof. The pharmaceutical preparation has an excellent intraocular pressure lowering effect and may be used as a therapeutic or preventive agen…
Who is the assignee on this patent?
Santen Pharmaceutical Co Ltd
What technology area does this patent fall under?
Primary CPC classification A61K31/444. Mapped technology areas include Human Necessities.
When was this patent published?
Publication date Tue Jan 15 2019 00:00:00 GMT+0000 (Coordinated Universal Time) (B2). Legal status and post-grant events are not shown on this page.
What related patents are in patentsdb?
We list 2 related publications on this page (citations in our corpus or others sharing the same primary CPC).